SCHEMBL5032591

SCHEMBL5032591

CS(=O)(=O)N1CCC(N(Cc2ccc(F)cc2F)c2ccc(C#N)c(Cl)c2)C1

nearest known ligand 0.82

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PGR P06401 20/20 0.82
CYP2C9 P11712 17/20 0.82
CYP2D6 P10635 15/20 0.82
KCNH2 Q12809 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3023924 1.00 PGR (0.82) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3017662 0.94 PGR (0.84) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3038626 0.93 PGR (0.80) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3033409 0.91 PGR (0.81) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3037226 0.91 PGR (0.82) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3024771 0.91 PGR (0.81) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3025793 0.90 PGR (0.78) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3035009 0.90 PGR (1.00) PGRCYP2C9CYP2D6KCNH2
SCHEMBL5030156 0.90 PGR (1.00) PGRCYP2C9CYP2D6KCNH2
SCHEMBL13218900 0.90 PGR (0.83) PGRCYP2C9CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954133-A2 PYRROLIDINEANILINES SMITHKLINE BEECHAM CORPORATION (US) 2008-08-13 EP claimed
WO-2007065093-A2 PYRROLIDINEANILINES SMITHKLINE BEECHAM CORPORATION (US) 2007-06-07 WO claimed