SCHEMBL5032599

SCHEMBL5032599

CS(=O)(=O)c1cccc(NC(=O)Oc2cnn3c(C(F)(F)F)cc(-c4ccc(C(F)(F)F)c(OCC(F)(F)F)c4)nc23)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.43
KDM4E B2RXH2 9/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 6/20 0.42
ALDH1A1 P00352 6/20 0.42
CYP3A4 P08684 3/20 0.42
GAA P10253 2/20 0.42
HSD17B10 Q99714 3/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
TSHR P16473 3/20 0.40
RXFP1 Q9HBX9 3/20 0.40
CASP1 P29466 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
CYP1A2 P05177 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CASP7 P55210 1/20 0.39
POLB P06746 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5036085 0.95 THRB (0.44) THRBKDM4EKMT2AMEN1LMNA
SCHEMBL5034925 0.91 KDM4E (0.48) THRBKDM4EKMT2AMEN1LMNA
SCHEMBL5041513 0.90 KDM4E (0.43) THRBKDM4EKMT2AMEN1LMNA
SCHEMBL5041410 0.90 KDM4E (0.43) THRBKDM4EKMT2AMEN1LMNA
SCHEMBL5036058 0.90 KDM4E (0.43) THRBKDM4EKMT2AMEN1LMNA
SCHEMBL5048295 0.89 THRB (0.54) THRBKDM4EKMT2AMEN1LMNA
SCHEMBL5041368 0.88 THRB (0.43) THRBKDM4EKMT2AMEN1LMNA
SCHEMBL5032624 0.87 KDM4E (0.44) THRBKDM4EKMT2AMEN1LMNA
SCHEMBL5035013 0.87 KDM4E (0.46) THRBKDM4EKMT2AMEN1LMNA
SCHEMBL5032652 0.86 KDM4E (0.44) THRBKDM4EKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed