SCHEMBL5032629

SCHEMBL5032629

O=C(Nc1cccc(S(=O)(=O)NCc2ccccc2)c1)Oc1cnn2c(C(F)F)cc(-c3ccc(C(F)(F)F)cc3)nc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.50
KDM4E B2RXH2 4/20 0.48
KMT2A Q03164 2/20 0.48
HTT P42858 1/20 0.48
POLB P06746 2/20 0.44
TP53 P04637 2/20 0.44
NAMPT P43490 1/20 0.42
NPY5R Q15761 1/20 0.42
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
RAB9A P51151 1/20 0.41
MAPT P10636 3/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
RECQL P46063 1/20 0.40
MGLL Q99685 1/20 0.40
IDH2 P48735 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5041326 0.91 MAPK1 (0.49) MAPK1KDM4EKMT2AHTTPOLB
SCHEMBL5035052 0.91 KDM4E (0.51) MAPK1KDM4EKMT2AHTTPOLB
SCHEMBL5039196 0.91 HPGD (0.45) MAPK1KDM4EHTTPOLBNAMPT
SCHEMBL5041572 0.91 MAPK1 (0.47) MAPK1KDM4EKMT2AHTTPOLB
SCHEMBL5035307 0.91 KDM4E (0.50) MAPK1KDM4EKMT2AHTTPOLB
SCHEMBL5039193 0.91 MAPK1 (0.49) MAPK1KDM4EKMT2AHTTPOLB
SCHEMBL5035000 0.90 KDM4E (0.49) MAPK1KDM4EKMT2AHTTPOLB
SCHEMBL5035008 0.89 KDM4E (0.51) MAPK1KDM4EKMT2AHTTPOLB
SCHEMBL5035072 0.89 KDM4E (0.54) MAPK1KDM4EKMT2AHTTPOLB
SCHEMBL5039123 0.89 MAPK1 (0.46) MAPK1KDM4EKMT2AHTTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed