SCHEMBL5041572

SCHEMBL5041572

O=C(Nc1cccc(S(=O)(=O)NCc2ccccn2)c1)Oc1cnn2c(C(F)F)cc(-c3ccc(C(F)(F)F)cc3)nc12

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.47
KDM4E B2RXH2 3/20 0.46
KMT2A Q03164 2/20 0.46
HTT P42858 1/20 0.46
MAPT P10636 3/20 0.42
TP53 P04637 2/20 0.41
POLB P06746 2/20 0.41
ALDH1A1 P00352 3/20 0.39
MCL1 Q07820 1/20 0.39
SYK P43405 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KIF18A Q8NI77 1/20 0.38
LMNA P02545 2/20 0.38
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5041331 0.91 HPGD (0.41) MAPK1KDM4EHTTMAPTALDH1A1
SCHEMBL5032629 0.91 MAPK1 (0.50) MAPK1KDM4EKMT2AHTTMAPT
SCHEMBL5044774 0.89 MAPK1 (0.56) MAPK1KDM4EKMT2AHTTMAPT
SCHEMBL5039193 0.89 MAPK1 (0.49) MAPK1KDM4EKMT2AHTTMAPT
SCHEMBL5041326 0.88 MAPK1 (0.49) MAPK1KDM4EKMT2AHTTMAPT
SCHEMBL5035052 0.88 KDM4E (0.51) MAPK1KDM4EKMT2AHTTMAPT
SCHEMBL5035307 0.88 KDM4E (0.50) MAPK1KDM4EKMT2AHTTMAPT
SCHEMBL5035000 0.87 KDM4E (0.49) MAPK1KDM4EKMT2AHTTMAPT
SCHEMBL5035008 0.86 KDM4E (0.51) MAPK1KDM4EKMT2AHTTMAPT
SCHEMBL5035072 0.86 KDM4E (0.54) MAPK1KDM4EKMT2AHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed