SCHEMBL5040333

SCHEMBL5040333

COc1ccc2c(C)cc(=O)n(CCN3CCC(N(Cc4ccc5c(c4)OCCO5)C(=O)O)CC3)c2c1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.58
HTR1A P08908 1/20 0.43
SLC6A4 P31645 1/20 0.43
OPRM1 P35372 2/20 0.42
LMNA P02545 5/20 0.42
THRB P10828 1/20 0.40
TP53 P04637 2/20 0.40
UBE2M P61081 1/20 0.40
DCUN1D1 Q96GG9 1/20 0.40
CNR2 P34972 1/20 0.39
MCHR1 Q99705 1/20 0.39
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2793478 0.94 KCNH2 (0.51) KCNH2HTR1ASLC6A4OPRM1LMNA
SCHEMBL2797923 0.93 KCNH2 (0.50) KCNH2OPRM1LMNATHRBTP53
SCHEMBL2798542 0.92 KCNH2 (0.49) KCNH2HTR1ASLC6A4OPRM1LMNA
SCHEMBL2797675 0.92 KCNH2 (0.49) KCNH2OPRM1LMNATHRBTP53
SCHEMBL2796266 0.91 KCNH2 (0.53) KCNH2HTR1ASLC6A4OPRM1LMNA
SCHEMBL5039995 0.90 KCNH2 (0.48) KCNH2HTR1ASLC6A4OPRM1LMNA
SCHEMBL2794337 0.90 KCNH2 (0.47) KCNH2HTR1ASLC6A4OPRM1LMNA
SCHEMBL5036618 0.90 KCNH2 (0.47) KCNH2HTR1ASLC6A4OPRM1LMNA
SCHEMBL5040901 0.89 THRB (0.46) KCNH2OPRM1LMNATHRBTP53
SCHEMBL5042261 0.89 KCNH2 (0.48) KCNH2HTR1ASLC6A4OPRM1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468743-A1 Nitrogen-containing bicyclic compounds useful as antibacterial agents Toyama Chemical Co., Ltd. (JP) 2012-06-27 EP disclosed
EP-1900732-A1 NOVEL NITROGENATED HETEROCYCLIC COMPOUND AND SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2008-03-19 EP disclosed