SCHEMBL5040977

SCHEMBL5040977

CS(=O)(=O)c1ccc(OC(F)(F)F)c(C(=O)N2CCN(c3ccc(C#N)cc3)CC2)c1

nearest known ligand 0.77

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 20/20 0.77
KCNH2 Q12809 7/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5047534 0.88 SLC6A9 (0.78) SLC6A9KCNH2
SCHEMBL5133024 0.87 SLC6A9 (0.79) SLC6A9KCNH2
SCHEMBL5042002 0.87 SLC6A9 (0.82) SLC6A9KCNH2
SCHEMBL4433638 0.87 SLC6A9 (1.00) SLC6A9KCNH2
SCHEMBL5038533 0.87 SLC6A9 (0.60) SLC6A9KCNH2
SCHEMBL5040959 0.87 SLC6A9 (0.59) SLC6A9KCNH2
SCHEMBL5046090 0.87 SLC6A9 (0.65) SLC6A9KCNH2
SCHEMBL5037772 0.86 SLC6A9 (0.71) SLC6A9KCNH2
SCHEMBL5042677 0.85 SLC6A9 (0.81) SLC6A9KCNH2
SCHEMBL4420159 0.85 SLC6A9 (0.69) SLC6A9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1867554-B Piperazine with ortho-substituted phenyl and its use as GLYT1 inhibitors HOFFMANN LA ROCHE 2011-07-06 CN disclosed
EP-1656361-B1 PIPERAZINE WITH OR-SUBSTITUTED PHENYL GROUP AND THEIR USE AS GLYT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed
CN-1867554-A Piperazine with ortho-substituted phenyl and its use as GLYT1 inhibitors HOFFMANN LA ROCHE (CH) 2006-11-22 CN disclosed