SCHEMBL5041740

SCHEMBL5041740

COCCN1CN(Cc2ccccn2)n2cc(CCCc3ccc(F)cc3F)c(=O)c(OCc3ccccc3)c2C1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KDM1A O60341 1/20 0.32
ABCB1 P08183 1/20 0.31
ABCC1 P33527 1/20 0.31
ABCG2 Q9UNQ0 1/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
FPR1 P21462 2/20 0.30
FPR2 P25090 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
CASP1 P29466 1/20 0.30
CYP2C19 P33261 1/20 0.30
CASP7 P55210 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4162790 0.86 KDM1A (0.34) KDM1AALDH1A1HPGDSMN1; SMN2CYP1A2
SCHEMBL8933626 0.86 MEN1 (0.40) MEN1KMT2A
SCHEMBL8211552 0.84 KDM1A (0.34) KDM1A
SCHEMBL8987614 0.80 MEN1 (0.42) MEN1KMT2A
SCHEMBL4165486 0.79 KDM1A (0.35) KDM1AALDH1A1HPGDCYP1A2CYP3A4
SCHEMBL4167513 0.78 MEN1 (0.34) MEN1KMT2A
SCHEMBL8933396 0.76 KCNA5 (0.41)
SCHEMBL8933329 0.76
SCHEMBL19158191 0.74 BRD4 (0.32) KDM1AALDH1A1HPGDCYP1A2CYP3A4
SCHEMBL8933586 0.74 KCNA5 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1950212-A1 POLYCYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING INHIBITORY ACTIVITY ON HIV INTEGRASE Shionogi Co., Ltd. (JP) 2008-07-30 EP disclosed