SCHEMBL8211552

SCHEMBL8211552

COCCN1CN(CCN(C)C(C)=O)n2cc(CCCc3ccc(F)cc3F)c(=O)c(OCc3ccccc3)c2C1=O

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.34
BCHE P06276 3/20 0.31
HTR2A P28223 1/20 0.31
FFAR1 O14842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4162790 0.87 KDM1A (0.34) KDM1ABCHE
SCHEMBL4167513 0.84 MEN1 (0.34)
SCHEMBL5041740 0.84 MEN1 (0.35) KDM1A
SCHEMBL8933396 0.79 KCNA5 (0.41)
SCHEMBL4165486 0.78 KDM1A (0.35) KDM1ABCHE
SCHEMBL8933586 0.77 KCNA5 (0.41)
SCHEMBL4173647 0.75
SCHEMBL19158282 0.73 KDM1A (0.34) KDM1A
SCHEMBL8933626 0.73 MEN1 (0.40)
SCHEMBL19158191 0.72 BRD4 (0.32) KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188271-B2 Polycyclic carbamoylpyridone derivative having HIV integrase inhibitory activity SHIONOGI & CO., LTD. (JP) 2012-05-29 US disclosed