SCHEMBL5042013

SCHEMBL5042013

Cc1ccc(N2CCN(C(=O)c3cc(S(C)(=O)=O)ccc3OC(C)C(F)(F)F)CC2)nc1

nearest known ligand 0.82

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 20/20 0.82
KCNH2 Q12809 7/20 0.82
SLC6A5 Q9Y345 2/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5037773 0.94 SLC6A9 (0.87) SLC6A9KCNH2SLC6A5
SCHEMBL5038277 0.90 SLC6A9 (0.81) SLC6A9KCNH2SLC6A5
SCHEMBL562797 0.90 SLC6A9 (1.00) SLC6A9KCNH2SLC6A5
SCHEMBL562110 0.90 SLC6A9 (0.81) SLC6A9KCNH2SLC6A5
SCHEMBL5040943 0.90 SLC6A9 (0.67) SLC6A9KCNH2SLC6A5
SCHEMBL5041835 0.88 SLC6A9 (0.78) SLC6A9KCNH2SLC6A5
SCHEMBL18502986 0.86 SLC6A9 (0.83) SLC6A9KCNH2SLC6A5
SCHEMBL5038042 0.84 SLC6A9 (0.84) SLC6A9KCNH2SLC6A5
SCHEMBL5042859 0.84 SLC6A9 (0.79) SLC6A9KCNH2SLC6A5
SCHEMBL5043601 0.84 SLC6A9 (0.85) SLC6A9KCNH2SLC6A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656361-B1 PIPERAZINE WITH OR-SUBSTITUTED PHENYL GROUP AND THEIR USE AS GLYT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed