SCHEMBL5042494

SCHEMBL5042494

CCCCCOc1ccc(F)c([C@H](OCC)C(=O)NCc2ccc(C#N)cc2)c1F

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FAAH O00519 3/20 0.41
MGLL Q99685 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
S1PR2 O95136 1/20 0.36
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
LPAR2 Q9HBW0 1/20 0.36
AKR1B1 P15121 1/20 0.36
EPHX2 P34913 1/20 0.35
VNN1 O95497 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6068735 0.86 EPHX2 (0.35) FAAHALDH1A1AKR1B1EPHX2VNN1
SCHEMBL5042490 0.86 EPHX2 (0.35) FAAHALDH1A1AKR1B1EPHX2VNN1
SCHEMBL5043807 0.84 EPHX2 (0.38) AKR1B1EPHX2VNN1
SCHEMBL5043811 0.84 EPHX2 (0.38) AKR1B1EPHX2VNN1
SCHEMBL5041935 0.84 EPHX2 (0.38) ALDH1A1AKR1B1EPHX2VNN1
SCHEMBL5041938 0.84 EPHX2 (0.38) ALDH1A1AKR1B1EPHX2VNN1
SCHEMBL5041085 0.83 PPARA (0.38) AKR1B1EPHX2VNN1
SCHEMBL5041087 0.83 PPARA (0.38) AKR1B1EPHX2VNN1
SCHEMBL5043438 0.82 EPHX2 (0.36) AKR1B1EPHX2VNN1
SCHEMBL5038100 0.82 AKR1B1 (0.37) AKR1B1EPHX2VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567498-B1 MANDELIC ACID DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-23 EP disclosed