Acetic Acid

Acetic Acid

SCHEMBL5042770

CC(=O)O.COC(C(=O)NCc1ccc(C(=N)N)cc1)c1c(F)ccc(Oc2cccnc2)c1F

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Acetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 1/20 0.40
F2 P00734 9/20 0.38
MASP2 O00187 1/20 0.38
MRGPRX1 Q96LB2 1/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
F7 P08709 3/20 0.37
F10 P00742 2/20 0.37
PRSS1 P07477 2/20 0.37
F3 P13726 2/20 0.36
ST14 Q9Y5Y6 1/20 0.36
PKM P14618 1/20 0.36
ADRA1B P35368 1/20 0.36
PROC P04070 1/20 0.36
CARM1 Q86X55 1/20 0.35
PRMT6 Q96LA8 1/20 0.35
LOX P28300 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5041562 0.89 F10 (0.45) PPARDF2MASP2MRGPRX1USP2
Hydrochloric Acid SCHEMBL5041559 0.89 F10 (0.45) PPARDF2MASP2MRGPRX1USP2
Acetic Acid SCHEMBL5043119 0.87 CARM1 (0.44) PPARDF2MASP2L3MBTL1F7
Hydrochloric Acid SCHEMBL5047274 0.85 MRGPRX1 (0.51) F2MRGPRX1USP2ALDH1A1NPSR1
Hydrochloric Acid SCHEMBL5047266 0.85 MRGPRX1 (0.51) F2MRGPRX1USP2ALDH1A1NPSR1
Acetic Acid SCHEMBL5041870 0.83 F10 (0.44) F2MASP2F7F10PRSS1
Hydrochloric Acid SCHEMBL5045176 0.79 F2 (0.44) F2MASP2MRGPRX1ALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL5045174 0.79 F2 (0.44) F2MASP2MRGPRX1ALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL5041613 0.79 CARM1 (0.49) F2MASP2F7F10PRSS1
Hydrochloric Acid SCHEMBL5041619 0.79 CARM1 (0.49) F2MASP2F7F10PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7129238-B2 Mandelic acid derivatives HOFFMANN-LA ROCHE INC. (US) 2006-10-31 US claimed
US-20040122057-A1 Novel mandelic acid derivatives HOFFMANN-LA ROCHE INC. 2004-06-24 US claimed
EP-1567498-B1 MANDELIC ACID DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-23 EP disclosed
US-7129238-B2 Mandelic acid derivatives HOFFMANN-LA ROCHE INC. (US) 2006-10-31 US disclosed
EP-1567498-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2005-08-31 EP disclosed
US-20040122057-A1 Novel mandelic acid derivatives HOFFMANN-LA ROCHE INC. 2004-06-24 US disclosed
WO-2004048335-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2004-06-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040122057-A1 Novel mandelic acid derivatives F7, F11, F9 PPARD 4571/4885F2 13/4885MASP2 370/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.