SCHEMBL5043687

SCHEMBL5043687

COc1ccccc1CNC(=O)Oc1nc2c(OC)ccc(N3CCOCC3)c2s1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 17/20 0.53
ADORA1 P30542 13/20 0.53
ADORA2B P29275 4/20 0.50
ADORA3 P0DMS8 2/20 0.50
ALDH1A1 P00352 1/20 0.50
MAPT P10636 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
KDM4E B2RXH2 1/20 0.49
GAA P10253 1/20 0.49
HSD17B10 Q99714 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5037316 0.92 ADORA2A (0.51) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5043776 0.88 ADORA2A (0.51) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5034125 0.86 ALDH1A1 (0.56) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL5034182 0.86 ADORA2A (0.49) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5034263 0.85 ADORA2A (0.52) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5036855 0.84 ADORA2A (0.51) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5037630 0.83 ADORA2A (0.51) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5041829 0.82 ADORA2A (0.56) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5038587 0.82 ADORA2A (0.63) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5037376 0.80 ADORA2A (0.56) ADORA2AADORA1ADORA2BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1450796-B1 BENZOTHIAZOLE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-04-09 EP claimed