SCHEMBL5044258

SCHEMBL5044258

CCCCCCCCCCCc1noc(-c2ccc(C([NH])CCc3ccc(Cl)c(Cl)c3)cc2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SPHK1 Q9NYA1 5/20 0.43
S1PR1 P21453 4/20 0.40
S1PR5 Q9H228 3/20 0.40
NPC1 O15118 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KDM4E B2RXH2 1/20 0.40
PKM P14618 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
SPHK2 Q9NRA0 6/20 0.39
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CHRM2 P08172 2/20 0.36
CHRM4 P08173 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5044385 1.00 SPHK1 (0.43) SPHK1S1PR1S1PR5NPC1ALDH1A1
SCHEMBL5039990 0.90 SPHK1 (0.41) SPHK1S1PR1S1PR5NPC1ALDH1A1
SCHEMBL5045522 0.87 NPC1 (0.41) SPHK1S1PR1S1PR5NPC1ALDH1A1
SCHEMBL5049037 0.87 NPC1 (0.41) SPHK1S1PR1S1PR5NPC1ALDH1A1
SCHEMBL5049461 0.85 SMN1; SMN2 (0.56) SPHK1S1PR1S1PR5NPC1ALDH1A1
SCHEMBL5044306 0.85 SMN1; SMN2 (0.56) SPHK1S1PR1S1PR5NPC1ALDH1A1
SCHEMBL5044844 0.81 SPHK1 (0.43) SPHK1S1PR1S1PR5NPC1ALDH1A1
SCHEMBL1855641 0.80 SPHK1 (0.50) SPHK1S1PR1NPC1ALDH1A1MAPT
SCHEMBL1854487 0.80 SPHK1 (0.50) SPHK1S1PR1NPC1ALDH1A1MAPT
SCHEMBL6824694 0.80 SPHK1 (0.42) SPHK1S1PR1S1PR5NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732534-B1 USE OF METHYLENE AMIDE DERIVATIVES IN CARDIOVASCULAR DISORDERS SERONO LAB (CH) 2008-07-23 EP claimed