SCHEMBL5044751

SCHEMBL5044751

CCCn1c(=O)c2c(nc(Cc3ccnnc3)n2CCN(CC)CCO)n(CCc2ccc(N)c(Cl)c2)c1=O.CCCn1c(=O)c2c(nc(Cc3ccnnc3)n2CCN(CC)CCO)n(CCc2ccc(N)cc2Cl)c1=O

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.48
ADORA2B P29275 9/20 0.33
ADORA2A P29274 5/20 0.32
ADORA3 P0DMS8 3/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TSHR P16473 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1334722 0.95 ADORA1 (0.49) ADORA1ADORA2BADORA2AADORA3ALDH1A1
SCHEMBL1333023 0.94 ADORA1 (0.50) ADORA1ADORA2BADORA2AADORA3ALDH1A1
SCHEMBL1333466 0.83 ADORA1 (0.47) ADORA1ADORA2BADORA2AADORA3ALDH1A1
SCHEMBL5044749 0.81 ADORA1 (0.42) ADORA1
SCHEMBL4176173 0.80 ADORA1 (0.62) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL1334330 0.80 ADORA1 (0.44) ADORA1ADORA2BADORA2AADORA3ALDH1A1
SCHEMBL1333191 0.78 ADORA1 (0.62) ADORA1ADORA2BADORA2AADORA3ALDH1A1
SCHEMBL4182302 0.78 ADORA1 (0.59) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL1333496 0.78 ADORA1 (0.56) ADORA1ADORA2BADORA2AADORA3ALDH1A1
SCHEMBL5653185 0.78 ADORA1 (0.43) ADORA1ADORA2BADORA2AADORA3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636229-A4 A1 ADENOSINE RECEPTOR ANTOGONISTS ENDACEA INC (US) 2008-07-30 EP claimed
EP-1636229-A2 A1 ADENOSINE RECEPTOR ANTOGONISTS Endacea, Inc. (US) 2006-03-22 EP claimed
WO-2005009343-A2 A1 ADENOSINE RECEPTOR ANTOGONISTS ENDACEA, INC. (US) 2005-02-03 WO claimed