SCHEMBL5045017

SCHEMBL5045017

c1cc(-c2ncc[nH]2)ncn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.45
MTOR P42345 1/20 0.45
ADK P55263 1/20 0.45
CCNT1 O60563 2/20 0.41
CCNA2 P20248 2/20 0.41
CDK2 P24941 2/20 0.41
CDK9 P50750 2/20 0.41
CCNA1 P78396 2/20 0.41
CDK5 Q00535 2/20 0.41
CDK5R1 Q15078 2/20 0.41
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPK14 Q16539 2/20 0.39
MAPK13 O15264 1/20 0.39
RAF1 P04049 1/20 0.39
MAPK9 P45984 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
KDM4E B2RXH2 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29446004 0.85 NISCH (0.55) NISCHMTORADKCCNT1CCNA2
SCHEMBL5491437 0.82
SCHEMBL2814353 0.74 HSP90AA1 (0.52) CCNT1CCNA2CDK2CDK9CCNA1
SCHEMBL30595872 0.74 HSP90AA1 (0.52) CCNT1CCNA2CDK2CDK9CCNA1
SCHEMBL30216772 0.73 NISCH (0.52) NISCHMTORADKALDH1A1MEN1
SCHEMBL28581729 0.73 NISCH (0.52) NISCHMTORADKALDH1A1MEN1
SCHEMBL16817999 0.72 MTOR (0.57) NISCHMTORADKALDH1A1MEN1
SCHEMBL117383 0.72 MTOR (0.57) NISCHMTORADKALDH1A1MEN1
SCHEMBL13910999 0.71 HSP90AA1 (0.50) CCNT1CCNA2CDK2CDK9CCNA1
SCHEMBL1688472 0.71 NISCH (0.68) NISCHMTORADKALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493876-B1 IMIDAZOLE DERIVATIVES AS CASEIN KINASE INHIBITORS PFIZER (US) 2014-02-12 EP disclosed
EP-1716150-B1 SUBSTITUTED HETEROCYCLIC COMPOUNDS AND METHODS OF USE AMGEN INC (US) 2008-04-23 EP disclosed
US-5716955-A Substituted imidazole compounds SMITHKLINE BEECHAM CORPORATION (US) 1998-02-10 US disclosed