SCHEMBL30595872

SCHEMBL30595872

c1cc(-c2ccncn2)ncn1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.52
CYP2D6 P10635 1/20 0.45
GRM5 P41594 2/20 0.44
MAPK9 P45984 4/20 0.41
MAPK14 Q16539 3/20 0.41
MAPK11 Q15759 2/20 0.41
MAPK13 O15264 1/20 0.41
RAF1 P04049 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK10 P53779 2/20 0.40
CCNT1 O60563 2/20 0.40
CCNA2 P20248 2/20 0.40
CDK2 P24941 2/20 0.40
CDK9 P50750 2/20 0.40
CCNA1 P78396 2/20 0.40
CDK5 Q00535 2/20 0.40
CDK5R1 Q15078 2/20 0.40
LATS1 O95835 1/20 0.40
LATS2 Q9NRM7 1/20 0.40
GSK3B P49841 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2814353 1.00 HSP90AA1 (0.52) HSP90AA1CYP2D6GRM5MAPK9MAPK14
SCHEMBL10402322 0.94 HSP90AA1 (0.48) HSP90AA1CYP2D6GRM5MAPK9MAPK14
SCHEMBL13910999 0.90 HSP90AA1 (0.50) HSP90AA1CYP2D6GRM5MAPK9MAPK14
SCHEMBL3107817 0.87 LMNA (0.44) HSP90AA1CYP2D6GRM5MAPK9MAPK14
SCHEMBL9903935 0.85 CYP2D6 (0.60) HSP90AA1CYP2D6GRM5MAPK9MAPK14
SCHEMBL4294864 0.84 KDM4E (0.67) HSP90AA1GRM5MAPK9MAPK14MAPK11
SCHEMBL29394083 0.84 KDM4E (0.67) HSP90AA1GRM5MAPK9MAPK14MAPK11
SCHEMBL25295479 0.83 TP53 (0.48) HSP90AA1CYP2D6GRM5MAPK9MAPK14
SCHEMBL5989213 0.83 HSP90AA1 (0.44) HSP90AA1CYP2D6GRM5MAPK9MAPK14
SCHEMBL8499115 0.83 CYP2D6 (0.53) HSP90AA1CYP2D6GRM5MAPK9MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116710453-A Kinase inhibitors and uses thereof 璧辰医药技术股份有限公司 2023-09-05 CN disclosed