SCHEMBL5045776

SCHEMBL5045776

CSc1c(-c2ccccc2)nc2ccccc2c1C(=O)NCCc1ccccc1C#N

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.56
CYP2C19 P33261 2/20 0.56
TACR3 P29371 8/20 0.54
LMNA P02545 2/20 0.53
CYP2C9 P11712 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP3A4 P08684 2/20 0.43
GAA P10253 1/20 0.43
CYP1A2 P05177 1/20 0.43
TP53 P04637 1/20 0.42
DHODH Q02127 1/20 0.41
HPGD P15428 1/20 0.41
PTGFR P43088 2/20 0.41
HIF1A Q16665 1/20 0.40
TSHR P16473 1/20 0.40
PDE10A Q9Y233 1/20 0.40
TACR2 P21452 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5045996 0.87 LMNA (0.57) CYP2D6CYP2C19TACR3LMNACYP2C9
SCHEMBL4665580 0.87 LMNA (0.55) CYP2D6CYP2C19TACR3LMNACYP2C9
SCHEMBL4668727 0.86 LMNA (0.53) CYP2D6CYP2C19TACR3LMNACYP2C9
SCHEMBL4667328 0.86 LMNA (0.53) CYP2D6CYP2C19TACR3LMNACYP2C9
SCHEMBL4667842 0.84 TACR3 (0.56) TACR3LMNAALDH1A1CYP3A4HPGD
SCHEMBL4665602 0.84 LMNA (0.57) CYP2D6CYP2C19TACR3LMNACYP2C9
SCHEMBL4665569 0.84 TACR3 (0.56) CYP2D6CYP2C19TACR3LMNACYP2C9
SCHEMBL5041963 0.83 TACR3 (0.55) CYP2D6CYP2C19TACR3LMNACYP2C9
SCHEMBL5045721 0.83 LMNA (0.51) CYP2D6CYP2C19TACR3LMNACYP2C9
SCHEMBL5042633 0.83 LMNA (0.56) CYP2D6CYP2C19TACR3LMNACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928835-A1 ALKYL SULFOXIDE QUINOLINES AS NK-3 RECEPTOR LIGANDS Astra Zeneca AB (SE) 2008-06-11 EP claimed
WO-2007035158-A1 ALKYL SULFOXIDE QUINOLINES AS NK-3 RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2007-03-29 WO claimed