SCHEMBL5046925

SCHEMBL5046925

CC(C)(C)OC(=O)n1c(-c2cc(OCc3ccncc3)c(Cl)c3c2C(=O)NC3)cc2cc(CN3CCCCC3)ccc21

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 6/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GPR119 Q8TDV5 1/20 0.34
HRH3 Q9Y5N1 9/20 0.33
PREP P48147 1/20 0.33
ATR Q13535 1/20 0.32
ATRIP Q8WXE1 1/20 0.32
NR1H2 P55055 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3046674 0.92 MEN1 (0.34) TBK1MEN1KMT2ANR1H2
SCHEMBL3046394 0.90 NR1H2 (0.33) TBK1HRH3ATRATRIPNR1H2
SCHEMBL3037182 0.90 ACHE (0.37) TBK1MEN1KMT2ANR1H2
SCHEMBL3046302 0.89 NR1H2 (0.38) TBK1ATRATRIPNR1H2
SCHEMBL3044037 0.88 ABCB1 (0.36)
SCHEMBL3044239 0.87 DRD4 (0.34) TBK1ATRATRIPNR1H2
SCHEMBL3051382 0.87 NR1H2 (0.36) TBK1ATRATRIPNR1H2
SCHEMBL3044187 0.87 ATR (0.33) TBK1ATRATRIPNR1H2
SCHEMBL3043648 0.87 ATR (0.33) TBK1ATRATRIPNR1H2
SCHEMBL3159224 0.87 HRH3 (0.39) TBK1HRH3ATRATRIP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed