SCHEMBL5046934

SCHEMBL5046934

CC(C)(C)OC(=O)n1c(-c2ccc(Cl)c3c2C(=O)NC3)cc2cc(C(N)CC(O)c3ccccc3)ccc21

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.37
CREBBP Q92793 1/20 0.37
NR1H2 P55055 18/20 0.36
NR1H3 Q13133 3/20 0.34
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3835087 0.85 BRD4 (0.34) BRD4CREBBPNR1H2NR1H3
SCHEMBL3033397 0.85 PLA2G1B (0.40) BRD4CREBBPNR1H2NR1H3
SCHEMBL5050608 0.84 BRD4 (0.35) BRD4CREBBPNR1H2NR1H3CA12
SCHEMBL3034386 0.82 BRD4 (0.51) BRD4CREBBPNR1H2NR1H3CA12
SCHEMBL3044227 0.81 BRD4 (0.39) BRD4CREBBPNR1H2NR1H3CA12
SCHEMBL3046659 0.81 NR1H2 (0.44) BRD4CREBBPNR1H2NR1H3
SCHEMBL3044633 0.80 NR1H2 (0.41) BRD4CREBBPNR1H2NR1H3
SCHEMBL3043890 0.79 BRD4 (0.38) BRD4CREBBPNR1H2NR1H3CA12
SCHEMBL3041891 0.78 NR1H2 (0.38) BRD4CREBBPNR1H2NR1H3
SCHEMBL3047590 0.78 NR1H2 (0.45) BRD4CREBBPNR1H2NR1H3CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed