SCHEMBL5047564

SCHEMBL5047564

CC(C)Oc1ccc(C(N)=O)cc1C(=O)N1CCN(c2ccc(C(F)(F)F)cc2C#N)CC1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 17/20 0.52
KCNH2 Q12809 8/20 0.51
SLC6A5 Q9Y345 3/20 0.43
ACACB O00763 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
ALOX12 P18054 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTT P42858 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CHRM4 P08173 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5041780 0.88 SLC6A9 (0.63) SLC6A9KCNH2SLC6A5CYP3A4CYP2C9
SCHEMBL4423788 0.85 SLC6A9 (0.73) SLC6A9KCNH2SLC6A5
SCHEMBL5045531 0.84 SLC6A9 (0.71) SLC6A9KCNH2SLC6A5
SCHEMBL5041433 0.82 SLC6A9 (0.73) SLC6A9KCNH2SLC6A5
SCHEMBL5047631 0.80 SLC6A9 (0.50) SLC6A9KCNH2
SCHEMBL5047807 0.79 SLC6A9 (0.58) SLC6A9KCNH2SLC6A5
SCHEMBL5038209 0.78 SLC6A9 (0.75) SLC6A9KCNH2SLC6A5HTTL3MBTL1
SCHEMBL4423405 0.76 SLC6A9 (0.64) SLC6A9KCNH2SLC6A5
SCHEMBL4425004 0.76 SLC6A9 (0.70) SLC6A9KCNH2SLC6A5
SCHEMBL5037700 0.76 SLC6A9 (0.54) SLC6A9KCNH2SLC6A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656361-B1 PIPERAZINE WITH OR-SUBSTITUTED PHENYL GROUP AND THEIR USE AS GLYT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed