SCHEMBL5047896

SCHEMBL5047896

COc1ccc(F)c(C(OC)C(=O)NCc2ccc(C(=N)N)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
F2 P00734 8/20 0.49
ST14 Q9Y5Y6 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.42
KLKB1 P03952 1/20 0.42
ALDH1A1 P00352 2/20 0.41
PRSS1 P07477 3/20 0.41
PRSS2 P07478 1/20 0.41
PRSS3 P35030 1/20 0.41
PKM P14618 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
F10 P00742 3/20 0.41
F7 P08709 2/20 0.41
PLAU P00749 1/20 0.40
PLAT P00750 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5047899 1.00 F2 (0.49) F2ST14L3MBTL1KLKB1ALDH1A1
Hydrochloric Acid SCHEMBL5041642 0.99 F2 (0.49) F2ST14L3MBTL1KLKB1ALDH1A1
Hydrochloric Acid SCHEMBL5041649 0.99 F2 (0.49) F2ST14L3MBTL1KLKB1ALDH1A1
SCHEMBL5042056 0.92 F2 (0.49) F2ST14L3MBTL1KLKB1ALDH1A1
SCHEMBL5042049 0.92 F2 (0.49) F2ST14L3MBTL1KLKB1ALDH1A1
Hydrochloric Acid SCHEMBL5045900 0.91 F2 (0.49) F2ST14L3MBTL1KLKB1ALDH1A1
Hydrochloric Acid SCHEMBL5045897 0.91 F2 (0.49) F2ST14L3MBTL1KLKB1ALDH1A1
SCHEMBL5041859 0.88 PKM (0.49) F2ST14KLKB1PRSS1PKM
SCHEMBL5041852 0.88 PKM (0.49) F2ST14KLKB1PRSS1PKM
Hydrochloric Acid SCHEMBL5047289 0.88 PKM (0.48) F2ST14KLKB1PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567498-B1 MANDELIC ACID DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-23 EP disclosed
EP-1567498-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2005-08-31 EP disclosed
WO-2004048335-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2004-06-10 WO disclosed