SCHEMBL5048276

SCHEMBL5048276

CC(C)(C)OC(=O)n1c(-c2ccc(Cl)c3c2C(=O)NC3)cc2cc(CN3CCCC(O)C3)ccc21

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.36
HTT P42858 1/20 0.36
ROCK2 O75116 1/20 0.35
BRD4 O60885 1/20 0.34
CREBBP Q92793 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MCHR1 Q99705 5/20 0.34
PDGFRB P09619 3/20 0.34
KDR P35968 3/20 0.34
LTA4H P09960 2/20 0.33
GRM2 Q14416 1/20 0.33
NR1H2 P55055 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
PARP1 P09874 1/20 0.33
PARP2 Q9UGN5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3039410 0.93 PDGFRB (0.37) HTTROCK2BRD4CREBBPALDH1A1
SCHEMBL3040224 0.92 PDE2A (0.38) PDE2AROCK2BRD4CREBBPNR1H2
SCHEMBL3038085 0.91 KDM4E (0.37) PDE2ABRD4CREBBPALDH1A1PDGFRB
SCHEMBL3047029 0.91 NR1H2 (0.37) BRD4CREBBPNR1H2PARP1
SCHEMBL3047413 0.90 NR1H2 (0.36) BRD4CREBBPNR1H2
SCHEMBL3044252 0.88 BRD4 (0.36) BRD4CREBBPALDH1A1NR1H2GPR119
SCHEMBL3037652 0.88 BRD4 (0.38) BRD4CREBBPALDH1A1NR1H2GPR119
SCHEMBL3043652 0.87 HSP90AA1 (0.37) BRD4CREBBPALDH1A1NR1H2GPR119
SCHEMBL3047734 0.87 VEGFA (0.40) NR1H2GPR119
SCHEMBL3048885 0.86 GPR119 (0.37) BRD4CREBBPALDH1A1PDGFRBKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed