SCHEMBL5048686

SCHEMBL5048686

N#[N+]c1ccc2ccsc2c1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.33
DYRK1A Q13627 1/20 0.31
MRGPRX4 Q96LA9 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5048601 0.83 CYP2A6 (0.46) CYP2A6DYRK1A
SCHEMBL8238127 0.79 CYP2A6 (0.33) CYP2A6DYRK1AMRGPRX4SLC6A2SLC6A4
SCHEMBL13742552 0.70 DYRK1A (0.48) CYP2A6DYRK1AMRGPRX4SLC6A2SLC6A4
SCHEMBL164774 0.69 CYP2A6 (0.50) CYP2A6DYRK1A
SCHEMBL18725843 0.67 CYP2A6 (0.36) CYP2A6DYRK1AMRGPRX4SLC6A2SLC6A4
SCHEMBL276241 0.67 CYP2A6 (0.41) CYP2A6DYRK1AMRGPRX4SLC6A2SLC6A4
SCHEMBL19914470 0.67 CYP2A6 (0.36) CYP2A6DYRK1AMRGPRX4SLC6A2SLC6A4
SCHEMBL422225 0.67 CYP2A6 (0.48) CYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL911044 0.67 ESR1 (0.44) CYP2A6MRGPRX4SLC6A2SLC6A4SLC6A3
SCHEMBL405354 0.67 CYP2A6 (0.41) CYP2A6DYRK1AMRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008062216-A1 ELECTRODE ISIS INNOVATION LIMITED (GB) 2008-05-29 WO disclosed