SCHEMBL5049246

SCHEMBL5049246

NC1(C(=O)O)CCC(C(F)(F)F)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 8/20 0.47
GRM2 Q14416 5/20 0.47
GRM3 Q14832 5/20 0.47
CYP1A2 P05177 4/20 0.47
CYP2C19 P33261 3/20 0.47
ALOX15 P16050 3/20 0.47
GRM8 O00222 3/20 0.47
GRM6 O15303 3/20 0.47
TDP1 Q9NUW8 2/20 0.47
LMNA P02545 1/20 0.47
GRM5 P41594 1/20 0.47
MTOR P42345 1/20 0.47
GRM1 Q13255 1/20 0.47
PLCB1 Q9NQ66 1/20 0.47
TSHR P16473 1/20 0.47
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2351634 0.98 GRM4 (0.46) GRM4GRM2GRM3CYP1A2CYP2C19
SCHEMBL4601909 0.79 GRM4 (0.47) GRM4GRM2GRM3CYP1A2CYP2C19
SCHEMBL4601083 0.79 GRM4 (0.47) GRM4GRM2GRM3CYP1A2CYP2C19
SCHEMBL1814154 0.77 NPSR1 (0.32) GRM4GRM2GRM3CYP1A2CYP2C19
SCHEMBL1814156 0.77 NPSR1 (0.32) GRM4GRM2GRM3CYP1A2CYP2C19
SCHEMBL31284547 0.77 ARG1 (0.46) GRM4GRM2GRM3CYP1A2CYP2C19
SCHEMBL1809492 0.77 NPSR1 (0.32) GRM4GRM2GRM3CYP1A2CYP2C19
SCHEMBL31231756 0.77 ARG1 (0.46) GRM4GRM2GRM3CYP1A2CYP2C19
SCHEMBL23882340 0.77 APP (0.32) CYP2C9
SCHEMBL12461686 0.77 APP (0.32) CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1220841-B1 TRIFLUOROMETHYL-SUBSTITUTED SPIROCYCLIC KETOENOLS BAYER CROPSCIENCE AG (DE) 2011-07-20 EP disclosed
US-7368424-B2 Acylated nonadepsipeptides AICURIS GMBH & CO. KG (DE) 2008-05-06 US disclosed
US-6861391-B1 Trifluoromethyl-substituted spirocyclic ketoenols BAYER AKTIENGESELLSCHAFT (DE) 2005-03-01 US disclosed