SCHEMBL5049313

SCHEMBL5049313

COc1cc(N2CCN(C(=O)C(C)C(C)N(C(=O)C(F)(F)F)c3ccccc3)CC2)c(Cl)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.45
KMT2A Q03164 2/20 0.41
LMNA P02545 5/20 0.41
MAPT P10636 3/20 0.41
NPY2R P49146 4/20 0.40
ALDH1A1 P00352 3/20 0.39
CNR1 P21554 1/20 0.39
MC4R P32245 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
RBP4 P02753 1/20 0.38
POLB P06746 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4508912 0.89 NPSR1 (0.45) NPSR1KMT2ALMNAMAPTNPY2R
Trifluoroacetic Acid SCHEMBL4508906 0.79 CCR1 (0.58) NPSR1KMT2ALMNAMAPTALDH1A1
SCHEMBL13606408 0.76 CCR1 (0.64) NPSR1KMT2ALMNAMAPTALDH1A1
SCHEMBL4501202 0.71 NPSR1 (0.48) NPSR1KMT2ALMNAMAPTALDH1A1
SCHEMBL4501206 0.71 NPSR1 (0.48) NPSR1KMT2ALMNAMAPTALDH1A1
Hydrochloric Acid SCHEMBL4502717 0.70 NPSR1 (0.48) NPSR1KMT2ALMNAMAPTALDH1A1
Hydrochloric Acid SCHEMBL4502722 0.70 NPSR1 (0.48) NPSR1KMT2ALMNAMAPTALDH1A1
SCHEMBL15164229 0.69 KMT2A (0.59) NPSR1KMT2ALMNAMAPTSMN1; SMN2
Trifluoroacetic Acid SCHEMBL5444922 0.68 LMNA (0.47) NPSR1KMT2ALMNAALDH1A1MC4R
Trifluoroacetic Acid SCHEMBL5444973 0.68 KMT2A (0.52) NPSR1KMT2ALMNAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973880-A1 PIPERAZINYL DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Brystol-Myers Squibb Company (US) 2008-10-01 EP disclosed
WO-2007087585-A1 PIPERAZINYL DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2007-08-02 WO disclosed