SCHEMBL5049609

SCHEMBL5049609

O=C(Cn1nc(-c2ccccc2)c(-c2ccc(Cl)cc2)n1)NN1CCOCC1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 6/20 0.50
SMN1; SMN2 Q16637 1/20 0.49
ALDH1A1 P00352 1/20 0.48
GAA P10253 1/20 0.48
ACHE P22303 1/20 0.47
BACE1 P56817 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
KDM5B Q9UGL1 2/20 0.47
LIPE Q05469 1/20 0.46
SLC2A2 P11168 1/20 0.45
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5050321 0.88 CNR2 (0.51) CNR1SMN1; SMN2GAAACHEBACE1
SCHEMBL3605027 0.75 SLC2A2 (0.58) GAACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL13307879 0.74 CNR1 (0.64) CNR1
SCHEMBL1787365 0.74 CYP3A4 (0.61) ALDH1A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL30795104 0.74 CYP3A4 (0.61) ALDH1A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4680489 0.74 CNR1 (0.60) CNR1SMN1; SMN2CYP2D6CYP2C9CYP2C19
SCHEMBL5050317 0.73 CNR1 (0.67) CNR1ALDH1A1KMT2A
SCHEMBL3604671 0.72 SLC2A2 (0.55) GAACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5359424 0.69 CNR1 (0.53) CNR1SMN1; SMN2CYP3A4CYP2C9CYP2C19
SCHEMBL6790329 0.69 SMN1; SMN2 (0.59) SMN1; SMN2ALDH1A1GAACYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1921072-A1 1,2,3-Triazole derivatives as cannabinoid-receptor modulators Laboratorios del Dr. Esteve S.A. (ES) 2008-05-14 EP claimed
EP-1921072-A1 1,2,3-Triazole derivatives as cannabinoid-receptor modulators Laboratorios del Dr. Esteve S.A. (ES) 2008-05-14 EP disclosed