SCHEMBL5050318

SCHEMBL5050318

Cc1ccccc1-c1cc2cnc(N(Cc3ccccc3)C3CCNCC3)nc2n(C2CCOCC2)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
CYP1A2 P05177 3/20 0.39
CYP3A4 P08684 3/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 3/20 0.39
USP2 O75604 2/20 0.39
CYP2D6 P10635 2/20 0.39
TSHR P16473 2/20 0.39
CASP1 P29466 2/20 0.39
CASP7 P55210 2/20 0.39
HSD17B10 Q99714 2/20 0.39
CDK4 P11802 4/20 0.39
CCND1 P24385 4/20 0.39
PIK3CA P42336 3/20 0.39
SLC6A4 P31645 6/20 0.38
SLC6A2 P23975 5/20 0.38
SLC6A3 Q01959 5/20 0.38
LCK P06239 1/20 0.37
MAPK14 Q16539 1/20 0.37
LYN P07948 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4040628 0.88 MAPK14 (0.40) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL3839596 0.86 MAPK14 (0.37) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4036260 0.85 MAPK14 (0.38) CDK4CCND1PIK3CALCKMAPK14
SCHEMBL5050315 0.85 PIK3CA (0.39) CYP2D6CDK4CCND1PIK3CASLC6A4
SCHEMBL4034535 0.84 PIK3CA (0.38) CDK4CCND1PIK3CASLC6A4SLC6A2
SCHEMBL5265811 0.84 ALDH1A1 (0.42) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL917926 0.80 MAPK14 (0.56) CDK4CCND1LCKMAPK14CDK6
SCHEMBL4139172 0.77 MAPK14 (0.53) CDK4CCND1LCKMAPK14CDK6
SCHEMBL3674451 0.76 MAPK14 (0.53) CYP1A2CYP3A4CYP2D6CDK4CCND1
SCHEMBL3671814 0.76 MAPK14 (0.53) CYP1A2CYP3A4CYP2D6CDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948164-A1 PHARMACEUTICAL COMPOSITIONS OF MUSCARINIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES, LTD. (IN) 2008-07-30 EP disclosed
WO-2007045979-A1 PHARMACEUTICAL COMPOSITIONS OF MUSCARINIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2007-04-26 WO disclosed