SCHEMBL5053296

SCHEMBL5053296

Cc1c(S(=O)(=O)Nc2ccc([N+](=O)[O-])cc2)cc(C(C)(C)C)c(O)c1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2L1 Q07817 1/20 0.53
MCL1 Q07820 1/20 0.53
ALDH1A1 P00352 5/20 0.46
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
KDM4E B2RXH2 2/20 0.46
HPGD P15428 2/20 0.46
CYP3A4 P08684 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.43
HTT P42858 2/20 0.43
GALR3 O60755 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CA2 P00918 2/20 0.42
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
GLRA3 O75311 1/20 0.42
GLRB P48167 1/20 0.42
MAPT P10636 3/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5057896 0.85 POLB (0.45) BCL2L1MCL1ALDH1A1MEN1KMT2A
SCHEMBL5061844 0.85 MCL1 (0.49) MCL1MEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL4114244 0.84 KMT2A (0.47) BCL2L1MCL1ALDH1A1MEN1KMT2A
SCHEMBL5067931 0.84 MCL1 (0.55) BCL2L1MCL1ALDH1A1MEN1KMT2A
SCHEMBL4113997 0.78 MEN1 (0.53) ALDH1A1MEN1KMT2AHPGDCYP3A4
SCHEMBL4137570 0.77 SMN1; SMN2 (0.42) MCL1ALDH1A1MEN1KMT2ATDP1
SCHEMBL4127131 0.76 KMT2A (0.49) ALDH1A1MEN1KMT2ASMN1; SMN2HTT
SCHEMBL4122654 0.74 MEN1 (0.46) ALDH1A1MEN1KMT2AHPGDTDP1
SCHEMBL4123794 0.74 MEN1 (0.46) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL4114911 0.73 KMT2A (0.50) ALDH1A1MEN1KMT2ATDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1890993-A2 BENZOIC ACID DERIVATIVES THAT ARE MODULATORS OR ANTAGONISTS OF GLYR AstraZeneca AB (SE) 2008-02-27 EP claimed
WO-2006121390-A2 BENZOIC ACID DERIVATIVES THAT ARE MODULATORS OR AGONISTS OF GLYR ASTRAZENECA AB (SE) 2006-11-16 WO claimed