SCHEMBL5067931

SCHEMBL5067931

Cc1c(S(=O)(=O)Nc2ccc([N+](=O)[O-])cc2)cc(C(C)C)c(O)c1C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 3/20 0.55
BCL2L1 Q07817 1/20 0.55
ALDH1A1 P00352 4/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
KDM4E B2RXH2 1/20 0.45
CYP3A4 P08684 1/20 0.45
HPGD P15428 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CA2 P00918 2/20 0.41
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
MAPT P10636 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
IDH1 O75874 2/20 0.41
POLB P06746 1/20 0.41
CYTH2 Q99418 1/20 0.40
HSD17B13 Q7Z5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4132975 0.84 KMT2A (0.44) MCL1BCL2L1ALDH1A1MEN1KMT2A
SCHEMBL5053296 0.84 BCL2L1 (0.53) MCL1BCL2L1ALDH1A1MEN1KMT2A
SCHEMBL4122107 0.73 PTGES (0.42) ALDH1A1MEN1KMT2AHPGDTDP1
SCHEMBL4128995 0.73 THRA (0.38) ALDH1A1MEN1KMT2ATDP1CA2
SCHEMBL29539746 0.71 MCL1 (1.00) MCL1BCL2L1
SCHEMBL18392406 0.71 MCL1 (1.00) MCL1BCL2L1
SCHEMBL5057896 0.70 POLB (0.45) MCL1BCL2L1ALDH1A1MEN1KMT2A
SCHEMBL5069803 0.70 BCL2L1 (0.60) MCL1BCL2L1ALDH1A1MEN1KMT2A
SCHEMBL5061844 0.69 MCL1 (0.49) MCL1MEN1KMT2AKDM4ECA2
SCHEMBL4115561 0.69 SMN1; SMN2 (0.52) BCL2L1ALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1890993-A2 BENZOIC ACID DERIVATIVES THAT ARE MODULATORS OR ANTAGONISTS OF GLYR AstraZeneca AB (SE) 2008-02-27 EP claimed
WO-2006121390-A2 BENZOIC ACID DERIVATIVES THAT ARE MODULATORS OR AGONISTS OF GLYR ASTRAZENECA AB (SE) 2006-11-16 WO claimed
EP-1890993-A2 BENZOIC ACID DERIVATIVES THAT ARE MODULATORS OR ANTAGONISTS OF GLYR AstraZeneca AB (SE) 2008-02-27 EP disclosed
WO-2006121390-A2 BENZOIC ACID DERIVATIVES THAT ARE MODULATORS OR AGONISTS OF GLYR ASTRAZENECA AB (SE) 2006-11-16 WO disclosed