SCHEMBL5053528

SCHEMBL5053528

COC(=O)C=CC1(C)CO1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.48
NFE2L2 Q16236 2/20 0.48
KEAP1 Q14145 1/20 0.48
ALDH1A1 P00352 4/20 0.35
ALOX15 P16050 1/20 0.35
RECQL P46063 1/20 0.35
HSD17B10 Q99714 1/20 0.35
KDM4E B2RXH2 2/20 0.34
MAPT P10636 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PRKCA P17252 4/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
TYR P14679 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32
TTR P02766 1/20 0.30
APP P05067 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5053526 1.00 HCAR2 (0.48) HCAR2NFE2L2KEAP1ALDH1A1ALOX15
SCHEMBL16040297 0.76 HCAR2 (0.40) HCAR2NFE2L2KEAP1ALDH1A1ALOX15
SCHEMBL16040296 0.76 HCAR2 (0.40) HCAR2NFE2L2KEAP1ALDH1A1ALOX15
SCHEMBL30936920 0.74 NFE2L2 (0.52) HCAR2NFE2L2KEAP1ALDH1A1ALOX15
SCHEMBL6060787 0.72 HCAR2 (0.40) HCAR2NFE2L2KEAP1ALDH1A1ALOX15
SCHEMBL6060792 0.72 HCAR2 (0.40) HCAR2NFE2L2KEAP1ALDH1A1ALOX15
SCHEMBL14677563 0.71 HCAR2 (0.48) HCAR2NFE2L2KEAP1ALDH1A1ALOX15
SCHEMBL8252913 0.71 HCAR2 (0.48) HCAR2NFE2L2KEAP1ALDH1A1ALOX15
SCHEMBL17518654 0.71 HCAR2 (0.43) HCAR2NFE2L2KEAP1ALDH1A1RECQL
SCHEMBL3883609 0.71 HCAR2 (0.43) HCAR2NFE2L2KEAP1ALDH1A1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080054171-A1 Target for Laser Desorption/Ionisation Mass Spectrometry PHYSIKALISCHES BURO STEINMULLER GMBH 2008-03-06 US claimed
WO-2007030849-A1 METHOD FOR DETECTING ORGANIC COMPOUNDS Austria Wirtschaftsservice Gesellschaft mit beschränkter Haftung (AT) 2007-03-22 WO claimed
US-20080054171-A1 Target for Laser Desorption/Ionisation Mass Spectrometry PHYSIKALISCHES BURO STEINMULLER GMBH 2008-03-06 US disclosed
WO-2007030849-A1 METHOD FOR DETECTING ORGANIC COMPOUNDS Austria Wirtschaftsservice Gesellschaft mit beschränkter Haftung (AT) 2007-03-22 WO disclosed
EP-1738397-A2 TARGET FOR LASER DESORPTION/IONISATION MASS SPECTROMETRY Physikalisches Büro Steinmüller GmbH (AT) 2007-01-03 EP disclosed
WO-2005096346-A2 TARGET FOR LASER DESORPTION/IONISATION MASS SPECTROMETRY PHYSIKALISCHES BÜRO STEINMÜLLER GMBH (AT) 2005-10-13 WO disclosed