Bromide

Bromide

SCHEMBL5053706

Br.Br.OB(O)Cc1ccccc1.c1cc(-c2ccncc2)ccn1

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 1/20 0.40
SLC6A4 known ✓ P31645 1/20 0.40
SLC6A3 known ✓ Q01959 1/20 0.40
NOTUM Q6P988 1/20 0.52
PRKCI P41743 1/20 0.46
ROCK2 O75116 5/20 0.45
ROCK1 Q13464 4/20 0.45
GSK3B P49841 3/20 0.45
CLK4 Q9HAZ1 3/20 0.45
RPS6KA5 O75582 2/20 0.45
MAP4K4 O95819 2/20 0.45
PRKACA P17612 2/20 0.45
MAPK1 P28482 2/20 0.45
GSK3A P49840 2/20 0.45
PRKX P51817 2/20 0.45
PRKG1 Q13976 2/20 0.45
PKN2 Q16513 2/20 0.45
SGK2 Q9HBY8 2/20 0.45
AKT1 P31749 2/20 0.45
PRKCG P05129 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyridine SCHEMBL1581039 0.88 CA1 (0.46) NOTUMMAPTLMNACA1CA2
SCHEMBL219668 0.81 CA1 (0.56) CA1CA2HSD17B10
SCHEMBL257595 0.77 CA1 (0.50) LMNACA1CA2RAB9A
Boric Acid SCHEMBL31391090 0.77 NOTUM (0.79) NOTUMPRKCIGSK3BPRKACAAKT1
Ethylene Glycol SCHEMBL8392416 0.74 CA1 (0.50) MAPTLMNACA1CA2
Dipyridyl SCHEMBL1897600 0.74 KDM4E (0.56) MAPK1MAPTLMNACA1CA2
Bromide SCHEMBL10968966 0.73 NOTUM (0.94) NOTUMGSK3BPRKACAAKT1RPS6KB1
SCHEMBL12030986 0.72 AGXT (0.50) PRKCICA1CA2
Pyridine SCHEMBL10928167 0.71 NOTUM (0.88) NOTUMGSK3BPRKACAAKT1RPS6KB1
SCHEMBL25377641 0.71 CA1 (0.46) LMNACA1CA2SLC6A2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960779-A2 OPTICAL DETERMINATION OF GLUCOSE UTILIZING BORONIC ACID ADDUCTS-II The Regents of the University of California (US) 2008-08-27 EP disclosed
WO-2007067743-A2 OPTICAL DETERMINATION OF GLUCOSE UTILIZING BORONIC ACID ADDUCTS-II THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2007-06-14 WO disclosed