SCHEMBL5059646

SCHEMBL5059646

CCc1c(Sc2ccc([N+](=O)[O-])cc2[N+](=O)[O-])cc(C(C)(C)C)c(O)c1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TXNRD1 Q16881 1/20 0.49
TXNRD3 Q86VQ6 1/20 0.49
TXNRD2 Q9NNW7 1/20 0.49
MAPT P10636 9/20 0.43
ALDH1A1 P00352 2/20 0.43
NPSR1 Q6W5P4 2/20 0.42
GAA P10253 2/20 0.42
HTT P42858 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
GALR3 O60755 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PSMD14 O00487 1/20 0.40
RAB9A P51151 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
GLRA3 O75311 1/20 0.39
GLRB P48167 1/20 0.39
LMNA P02545 2/20 0.39
FAAH O00519 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4121020 0.86 TXNRD1 (0.52) TXNRD1TXNRD3TXNRD2MAPTALDH1A1
SCHEMBL4122724 0.75 PDE7A (0.47) MAPTNPSR1GAAMEN1KMT2A
SCHEMBL4123964 0.73 SLC6A2 (0.44) MAPTALDH1A1NPSR1GAAHTT
SCHEMBL4121656 0.73 KMT2A (0.42) MAPTALDH1A1GAAHTTMEN1
SCHEMBL4122654 0.72 MEN1 (0.46) MAPTALDH1A1GAAHTTMEN1
SCHEMBL5059416 0.71 GLRA3 (0.43) GLRA3GLRBCA1CA2
SCHEMBL1032814 0.70 TXNRD1 (1.00) TXNRD1TXNRD3TXNRD2MAPTALDH1A1
SCHEMBL4128042 0.69 MEN1 (0.43) MAPTALDH1A1HTTMEN1KMT2A
SCHEMBL4113997 0.69 MEN1 (0.53) ALDH1A1HTTMEN1KMT2ASMN1; SMN2
SCHEMBL4122737 0.69 SMN1; SMN2 (0.43) MAPTALDH1A1GAAHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1890993-A2 BENZOIC ACID DERIVATIVES THAT ARE MODULATORS OR ANTAGONISTS OF GLYR AstraZeneca AB (SE) 2008-02-27 EP claimed
WO-2006121390-A2 BENZOIC ACID DERIVATIVES THAT ARE MODULATORS OR AGONISTS OF GLYR ASTRAZENECA AB (SE) 2006-11-16 WO claimed