SCHEMBL5064038

SCHEMBL5064038

CCOC(=O)c1cc(C#N)c(N2CCC2)nc1N(C)C

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.63
KDM4E B2RXH2 8/20 0.63
L3MBTL1 Q9Y468 4/20 0.63
LMNA P02545 1/20 0.63
HPGD P15428 1/20 0.63
TDP1 Q9NUW8 1/20 0.63
KMT2A Q03164 4/20 0.56
MEN1 O00255 3/20 0.56
MAPT P10636 1/20 0.56
MAPK1 P28482 1/20 0.53
HTT P42858 1/20 0.52
P2RY12 Q9H244 7/20 0.49
HSD17B10 Q99714 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5053551 0.97 ALDH1A1 (0.65) ALDH1A1KDM4EL3MBTL1LMNAHPGD
SCHEMBL4877133 0.88 P2RY12 (0.56) ALDH1A1KDM4EL3MBTL1LMNAHPGD
SCHEMBL4872829 0.85 P2RY12 (0.55) ALDH1A1KDM4EL3MBTL1LMNAHPGD
SCHEMBL5066024 0.81 ALDH1A1 (0.83) ALDH1A1KDM4EP2RY12NPSR1
SCHEMBL4875503 0.79 KDM4E (0.54) ALDH1A1KDM4EL3MBTL1LMNAHPGD
SCHEMBL4007118 0.78 ALDH1A1 (0.58) ALDH1A1KDM4EL3MBTL1LMNAHPGD
SCHEMBL4005299 0.78 ALDH1A1 (0.70) ALDH1A1KDM4EL3MBTL1LMNAHPGD
SCHEMBL4875182 0.77 P2RY12 (0.83) P2RY12
SCHEMBL30999840 0.76 ALDH1A1 (0.76) ALDH1A1KDM4EL3MBTL1LMNAHPGD
SCHEMBL3874439 0.76 ALDH1A1 (0.76) ALDH1A1KDM4EL3MBTL1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904474-A1 NEW PYRIDINE ANALOGUES AstraZeneca AB (SE) 2008-04-02 EP disclosed
WO-2007008140-A1 NEW PYRIDINE ANALOGUES ASTRAZENECA AB (SE) 2007-01-18 WO disclosed