SCHEMBL5065373

SCHEMBL5065373

CC(C)C(N)c1nc(C(=O)NC(c2nc(C(=O)NC(c3nc(C(=O)O)co3)C(C)C)co2)C(C)C)co1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
C3AR1 Q16581 17/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
PDE2A O00408 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL800524 0.89 C3AR1 (0.34) C3AR1HDAC1HDAC8HDAC6
SCHEMBL805184 0.79 HDAC1 (0.33) C3AR1HDAC1HDAC8HDAC6PDE2A
SCHEMBL801034 0.79 HDAC1 (0.42) C3AR1HDAC1HDAC8HDAC6
SCHEMBL800942 0.78 HDAC1 (0.33) C3AR1HDAC1HDAC8HDAC6
SCHEMBL805242 0.76 C3AR1 (0.31) C3AR1
SCHEMBL800480 0.74 C3AR1 (0.49) C3AR1
SCHEMBL25387512 0.74 HDAC1 (0.40) C3AR1HDAC1HDAC8HDAC6
SCHEMBL22636149 0.72 C3AR1 (0.37) C3AR1HDAC1HDAC8HDAC6
SCHEMBL22636152 0.72 C3AR1 (0.37) C3AR1HDAC1HDAC8HDAC6
SCHEMBL5512580 0.70 HDAC1 (0.41) HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009942-A1 HETEROAROMATIC-BASED PEPTIDE MACROCYCLES AS G-QUADRUPLEX LIGANDS CAMBRIDGE ENTERPRISE LTD. (GB) 2008-01-24 WO disclosed