SCHEMBL5065928

SCHEMBL5065928

Cc1ccc(C(=O)Nc2ccc(OC(=O)OCC(C(=O)O)(C(=O)O)c3ccccn3)cc2C(=O)N(C)C)c(-c2ccc(C(F)(F)F)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 4/20 0.41
NTRK2 Q16620 1/20 0.41
SORT1 Q99523 1/20 0.34
CASR P41180 1/20 0.34
OPRL1 P41146 1/20 0.34
F10 P00742 1/20 0.34
KDR P35968 2/20 0.33
TEK Q02763 2/20 0.33
MAPK14 Q16539 3/20 0.32
SMO Q99835 2/20 0.32
LIPE Q05469 1/20 0.32
LMNA P02545 1/20 0.32
PYGL P06737 1/20 0.32
PYGM P11217 1/20 0.32
AURKA O14965 1/20 0.32
ABL1 P00519 1/20 0.32
EGFR P00533 1/20 0.32
INSR P06213 1/20 0.32
LCK P06239 1/20 0.32
FES P07332 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14031657 0.93 NTRK1 (0.40) NTRK1NTRK2CASROPRL1F10
SCHEMBL5065162 0.87 NTRK1 (0.42) NTRK1NTRK2SORT1CASROPRL1
SCHEMBL5061890 0.82 MTTP (0.40) SMO
SCHEMBL5065207 0.82 NTRK1 (0.35) NTRK1NTRK2CASROPRL1F10
SCHEMBL5061956 0.82 F10 (0.36) NTRK1F10TRPV1
SCHEMBL5061900 0.81 MTTP (0.38) SMO
SCHEMBL5065208 0.80 CASR (0.31) NTRK1NTRK2CASRF10PTPN1
SCHEMBL5061983 0.79 TRPV1 (0.35) F10TRPV1
SCHEMBL5065185 0.79 LCK (0.39) NTRK1CASROPRL1F10KDR
SCHEMBL5066043 0.78 CASR (0.43) NTRK1NTRK2CASROPRL1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7432392-B2 Ester derivatives and medical use thereof JAPAN TOBACCO INC. (JP) 2008-10-07 US disclosed
US-20060205726-A1 Ester derivatives and medical use thereof JAPAN TOBACCO INC. (JP) 2006-09-14 US disclosed
EP-1669345-A1 ESTER DERIVATIVE AND MEDICINAL USE THEREOF JAPAN TOBACCO INC. (JP) 2006-06-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060205726-A1 Ester derivatives and medical use thereof MTTP, LIPC, CETP NTRK1 4115/4885NTRK2 3028/4885SORT1 898/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.