SCHEMBL5068898

SCHEMBL5068898

O=S(=O)(NCC1CCC(C#CCCCI)CC1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.43
CYP19A1 P11511 1/20 0.41
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
HDAC4 P56524 1/20 0.39
TGFBR1 P36897 1/20 0.39
USP30 Q70CQ3 1/20 0.39
MMP1 P03956 1/20 0.39
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
CYP2C9 P11712 1/20 0.38
CNR2 P34972 5/20 0.38
CNR1 P21554 2/20 0.38
PARG Q86W56 1/20 0.37
CA9 Q16790 1/20 0.37
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6529024 0.89 GBA1 (0.43) GBA1CYP19A1CA1CA2HDAC4
SCHEMBL5069078 0.81 LSS (0.53) GBA1TGFBR1KMT2AALDH1A1MEN1
SCHEMBL4803526 0.77 HTR2A (0.53) KMT2AALDH1A1MEN1HTR2C
SCHEMBL4803531 0.77 HTR2A (0.53) KMT2AALDH1A1MEN1HTR2C
SCHEMBL25252825 0.73 HTR2C (0.53) GBA1CYP19A1CA1CA2HDAC4
SCHEMBL5028418 0.72 KMT2A (0.70) GBA1CYP19A1MMP1KMT2AALDH1A1
SCHEMBL5028416 0.72 KMT2A (0.70) GBA1CYP19A1MMP1KMT2AALDH1A1
SCHEMBL7211522 0.72 USP30 (0.44) GBA1CYP19A1CA1CA2HDAC4
SCHEMBL7204569 0.70 GBA1 (0.46) GBA1CYP19A1CA1CA2HDAC4
SCHEMBL30700167 0.70 CYP19A1 (0.54) GBA1CYP19A1CA1CA2HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1311475-B1 AMINOCYCLOHEXANE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-08-06 EP disclosed