SCHEMBL5069415

SCHEMBL5069415

COCCCc1cc(CN(C(=O)C(CNC(=O)O)Cc2ccc(OCCOc3c(Cl)cc(C)cc3Cl)cc2)C2CC2)cc(OCc2ncccc2O)c1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.64
REN P00797 19/20 0.57
KCNH2 Q12809 10/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5069697 0.92 CYP3A4 (0.77) CYP3A4RENKCNH2
SCHEMBL4351586 0.90 CYP3A4 (0.66) CYP3A4RENKCNH2
SCHEMBL4349317 0.90 CYP3A4 (0.66) CYP3A4RENKCNH2
SCHEMBL4347867 0.90 CYP3A4 (0.68) CYP3A4RENKCNH2
SCHEMBL663978 0.88 CYP3A4 (0.67) CYP3A4RENKCNH2
SCHEMBL5071363 0.88 CYP3A4 (0.79) CYP3A4RENKCNH2
SCHEMBL4362212 0.86 CYP3A4 (0.71) CYP3A4RENKCNH2
SCHEMBL664368 0.86 CYP3A4 (0.71) CYP3A4RENKCNH2
SCHEMBL662715 0.86 CYP3A4 (0.70) CYP3A4RENKCNH2
SCHEMBL668325 0.85 CYP3A4 (0.64) CYP3A4RENKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910272-A1 RENIN INHIBITORS Merck Frosst Canada Ltd. (CA) 2008-04-16 EP disclosed
WO-2007009250-A1 RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2007-01-25 WO disclosed