SCHEMBL5069438

SCHEMBL5069438

Clc1c2ccccc2nn1-c1ccc(OCC2CCCN2I)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.46
GABRA1 P14867 1/20 0.39
GABRA2 P47869 1/20 0.39
CHRNB1 P11230 2/20 0.38
CHRNB2 P17787 2/20 0.38
CHRNB4 P30926 2/20 0.38
CHRNA3 P32297 2/20 0.38
CHRNA4 P43681 2/20 0.38
CHRNB3 Q05901 2/20 0.38
AXL P30530 1/20 0.36
MPO P05164 1/20 0.36
KCNH2 Q12809 1/20 0.35
MCHR1 Q99705 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9968590 0.82 LTA4H (0.56) ESR2KCNH2
SCHEMBL5069931 0.82 LTA4H (0.56) ESR2KCNH2
Hydrochloric Acid SCHEMBL3597194 0.81 LTA4H (0.55) ESR2KCNH2
Hydrochloric Acid SCHEMBL3598149 0.81 LTA4H (0.55) ESR2KCNH2
Hydrochloric Acid SCHEMBL3597192 0.81 LTA4H (0.55) ESR2KCNH2
SCHEMBL13436381 0.81 LTA4H (0.61) ESR2KCNH2
SCHEMBL3597992 0.80 LTA4H (0.44) ESR2
SCHEMBL3597998 0.80 LTA4H (0.44) ESR2
Hydrochloric Acid SCHEMBL3592985 0.80 LTA4H (0.60) ESR2KCNH2
Hydrochloric Acid SCHEMBL3592982 0.80 LTA4H (0.60) ESR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963276-A1 N-LINKED ARYL HETEROARYL INHIBITORS OF LTA4H FOR TREATING INFLAMMATION Decode Genetics EHF (IS) 2008-09-03 EP disclosed
WO-2007073405-A1 N-LINKED ARYL HETEROARYL INHIBITORS OF LTA4H FOR TREATING INFLAMMATION DECODE GENETICS EHF (IS) 2007-06-28 WO disclosed