SCHEMBL5071389

SCHEMBL5071389

CCCCN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Cc1c(-c2ccc(Cl)cc2)nc(-c2ccccc2)n1CCCC

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 5/20 0.42
C5AR1 P21730 1/20 0.40
TACR1 P25103 3/20 0.38
DHFR P00374 2/20 0.38
GPBAR1 Q8TDU6 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL650550 0.95 C5AR1 (0.44) CRHR1C5AR1TACR1TSHR
SCHEMBL5134817 0.93 CRHR1 (0.43) CRHR1C5AR1DHFR
SCHEMBL5137477 0.92 CRHR1 (0.43) CRHR1C5AR1DHFRTSHR
SCHEMBL647725 0.89 C5AR1 (0.41) CRHR1C5AR1TACR1TSHR
SCHEMBL5134950 0.89 C5AR1 (0.45) CRHR1C5AR1TSHR
SCHEMBL5135824 0.88 C5AR1 (0.44) CRHR1C5AR1TSHR
SCHEMBL5136524 0.88 C5AR1 (0.46) CRHR1C5AR1TSHR
SCHEMBL649523 0.87 MEN1 (0.46) CRHR1C5AR1TSHR
SCHEMBL5135207 0.87 C5AR1 (0.42) CRHR1C5AR1TSHR
SCHEMBL5135730 0.87 C5AR1 (0.41) CRHR1C5AR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed