SCHEMBL5073231

SCHEMBL5073231

C[N]C1CCC(CN2C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 4/20 0.49
ACHE P22303 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 6/20 0.46
HPGD P15428 3/20 0.46
KDM4E B2RXH2 3/20 0.46
GAA P10253 2/20 0.46
CYP3A4 P08684 1/20 0.46
ADRB2 P07550 3/20 0.44
ADRB1 P08588 3/20 0.44
ADRB3 P13945 3/20 0.44
KMT2A Q03164 1/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TRPA1 O75762 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1581709 0.87 CYP1B1 (0.59) CYP1B1ACHECYP1A2CYP2C9CYP2C19
SCHEMBL23439163 0.82 CYP1B1 (0.52) CYP1B1ACHECYP1A2CYP2C9CYP2C19
SCHEMBL19398815 0.82 CYP1B1 (0.52) CYP1B1ACHECYP1A2CYP2C9CYP2C19
SCHEMBL7583645 0.82 CYP1B1 (0.47) CYP1B1ACHECYP1A2CYP2C9CYP2C19
SCHEMBL7583648 0.82 CYP1B1 (0.47) CYP1B1ACHECYP1A2CYP2C9CYP2C19
Cyanide SCHEMBL27937317 0.82 CYP1B1 (0.55) CYP1B1ACHECYP1A2CYP2C9CYP2C19
SCHEMBL17268190 0.79 ACHE (0.55) CYP1B1ACHECYP1A2CYP2C9CYP2C19
SCHEMBL15537156 0.79 ACHE (0.55) CYP1B1ACHECYP1A2CYP2C9CYP2C19
SCHEMBL383479 0.79 CYP1B1 (0.52) CYP1B1ACHECYP1A2CYP2C9CYP2C19
SCHEMBL21598051 0.79 CYP1A2 (0.54) CYP1B1ACHECYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444235-B1 REVERSE-TURN MIMETICS AND METHOD RELATING THERETO CHOONGWAE PHARMA CORP (KR) 2008-06-11 EP disclosed