SCHEMBL5073458

SCHEMBL5073458

O=CCN1CCC(Nc2ccccc2Oc2ccc(Cl)cc2Cl)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 2/20 0.43
KCNH2 Q12809 1/20 0.42
LMNA P02545 3/20 0.42
MAPT P10636 2/20 0.42
KDM1A O60341 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD2 P14416 1/20 0.39
SLC6A12 P48065 1/20 0.39
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
BACE1 P56817 1/20 0.39
PLA2G1B P04054 1/20 0.38
ATG4B Q9Y4P1 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5071388 0.86 DRD2 (0.41) MCHR1SLC6A4KCNH2LMNAMEN1
SCHEMBL641135 0.81 MAPT (0.42) SLC6A2SLC6A4SLC6A3LMNAMAPT
SCHEMBL5073514 0.81 CHRM1 (0.46) MCHR1LMNAMAPTSIGMAR1MEN1
SCHEMBL642098 0.80 NPSR1 (0.52) SLC6A2SLC6A4SLC6A3LMNAMAPT
SCHEMBL641134 0.78 CNR1 (0.49) LMNAMEN1KMT2ACHRM1ACHE
SCHEMBL9965376 0.77 SMN1; SMN2 (0.50) SLC6A2SLC6A4SLC6A3LMNAMAPT
SCHEMBL9965435 0.77 CNR1 (0.49) LMNAMAPTMEN1KMT2ACHRM1
SCHEMBL640909 0.77 SLC6A4 (0.48) SLC6A2SLC6A4SLC6A3LMNAMAPT
SCHEMBL9965413 0.77 CNR1 (0.46) LMNAMAPTMEN1KMT2ACHRM1
SCHEMBL9965470 0.76 NPSR1 (0.49) LMNAMAPTMEN1KMT2ACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960347-A2 17-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 3 (17BETA-HSD3) INHIBITORS Sterix Limited (GB) 2008-08-27 EP disclosed
WO-2007003934-A2 17BETA-HYDR0XYSTER0ID DEHYDROGENASE TYPE 3 (17BETA-HSD3 ) INHIBITORS STERIX LIMITED (GB) 2007-01-11 WO disclosed