SCHEMBL5075012

SCHEMBL5075012

COc1cc(C(CC(C)C)=C(c2ccc(O)cc2)c2ccc(O)cc2)ccc1OCCN(C)C

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESRRB O95718 7/20 0.62
ESR1 P03372 11/20 0.46
ESRRG P62508 7/20 0.46
ESR2 Q92731 3/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
HIF1A Q16665 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
PLD2 O14939 1/20 0.46
PGR P06401 1/20 0.46
PLD1 Q13393 1/20 0.46
THRA P10827 1/20 0.44
THRB P10828 1/20 0.44
ESRRA P11474 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5075269 0.87 ESR1 (0.60) ESRRBESR1ESRRGESR2KDM4E
SCHEMBL5075821 0.85 THRA (0.53) ESRRBESR1ESRRGESR2KDM4E
SCHEMBL5075263 0.83 THRA (0.56) ESRRBESR1ESRRGESR2KDM4E
SCHEMBL4637955 0.82 ESR1 (0.60) ESRRBESR1ESRRGESR2KDM4E
SCHEMBL4637821 0.81 ESR1 (0.50) ESRRBESR1ESRRGESR2KDM4E
SCHEMBL5004320 0.79 ESR1 (0.52) ESRRBESR1ESRRGESR2KDM4E
SCHEMBL10016270 0.77 ESRRB (1.00) ESRRBESR1ESRRGESR2KDM4E
SCHEMBL20534069 0.77 ESRRB (1.00) ESRRBESR1ESRRGESR2KDM4E
SCHEMBL21294103 0.75 MAOB (0.65) KDM4EMEN1ALDH1A1KMT2ATHRA
SCHEMBL3813207 0.73 CYP19A1 (0.57) ESR1ESR2KDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951250-A2 CHEMICAL COMPOUNDS SmithKline Beecham Corporation (US) 2008-08-06 EP disclosed
WO-2007062151-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-31 WO disclosed