SCHEMBL508086

SCHEMBL508086

NCCCOc1ccc(-n2nc3ccccc3n2)c(O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
LMNA P02545 1/20 0.41
ESR1 P03372 2/20 0.39
CYP19A1 P11511 2/20 0.39
ESR2 Q92731 2/20 0.39
PDK2 Q15119 1/20 0.39
FGFR1 P11362 1/20 0.38
KDM4E B2RXH2 3/20 0.37
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
POLB P06746 1/20 0.35
HTT P42858 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.34
CYSLTR2 Q9NS75 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6474039 0.92 NPC1 (0.45) NPC1RAB9ALMNAFGFR1KDM4E
SCHEMBL8854056 0.90 NPC1 (0.44) NPC1RAB9ALMNAFGFR1KDM4E
SCHEMBL29463600 0.88 GPBAR1 (0.46) NPC1RAB9ALMNAFGFR1KDM4E
SCHEMBL7141357 0.88 GPBAR1 (0.46) NPC1RAB9ALMNAFGFR1KDM4E
SCHEMBL8913712 0.86 NPC1 (0.43) NPC1RAB9ALMNACYP19A1PDK2
SCHEMBL21145629 0.85 NPC1 (0.46) NPC1RAB9ALMNAPDK2FGFR1
SCHEMBL29510555 0.85 NPC1 (0.46) NPC1RAB9ALMNAPDK2FGFR1
SCHEMBL13370102 0.84 NR5A1 (0.50) NPC1RAB9ALMNAPDK2FGFR1
SCHEMBL5445426 0.84 NR5A1 (0.50) NPC1RAB9ALMNAPDK2FGFR1
SCHEMBL9744615 0.84 NR5A1 (0.50) NPC1RAB9ALMNAPDK2FGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104871036-B Method for making improved UV-absorbing ophthalmic lenses 诺华股份有限公司 2019-12-10 CN disclosed
EP-3542193-A1 METHOD FOR MAKING OPHTHALMIC LENSES Novartis AG (CH) 2019-09-25 EP disclosed
US-10338408-B2 Method for making improved UV-absorbing ophthalmic lenses NOVARTIS AG (CH) 2019-07-02 US disclosed
US-20180141293-A1 METHOD FOR MAKING OPHTHALMIC LENSES ALCON INC. (CH) 2018-05-24 US disclosed
EP-2598936-B1 METHOD FOR MAKING UV-ABSORBING OPHTHALMIC LENSES NOVARTIS AG (CH) 2017-11-01 EP disclosed
EP-2932314-B1 METHOD FOR MAKING IMPROVED UV-ABSORBING OPHTHALMIC LENSES NOVARTIS AG (CH) 2017-02-01 EP disclosed
EP-2766750-B1 METHOD FOR MAKING UV-ABSORBING OPHTHALMIC LENSES BY COATING NOVARTIS AG (CH) 2016-02-03 EP disclosed
EP-2932314-A1 METHOD FOR MAKING IMPROVED UV-ABSORBING OPHTHALMIC LENSES Novartis AG (CH) 2015-10-21 EP disclosed
US-9052439-B2 Method for making UV-absorbing ophthalmic lenses NOVARTIS AG (CH) 2015-06-09 US disclosed
US-9005700-B2 Method for making UV-absorbing ophthalmic lenses NOVARTIS AG (CH) 2015-04-14 US disclosed
EP-2766750-A1 METHOD FOR MAKING UV-ABSORBING OPHTHALMIC LENSES BY COATING Novartis AG (CH) 2014-08-20 EP disclosed
US-20140178595-A1 Method for Making Improved UV-Absorbing Ophthalmic Lenses NOVARTIS AG (CH) 2014-06-26 US disclosed
WO-2014095690-A1 METHOD FOR MAKING IMPROVED UV-ABSORBING OPHTHALMIC LENSES NOVARTIS AG (CH) 2014-06-26 WO disclosed
EP-2598936-A1 METHOD FOR MAKING UV-ABSORBING OPHTHALMIC LENSES Novartis AG (CH) 2013-06-05 EP disclosed
WO-2013055746-A1 METHOD FOR MAKING UV-ABSORBING OPHTHALMIC LENSES BY COATING NOVARTIS AG (CH) 2013-04-18 WO disclosed
US-20130095235-A1 METHOD FOR MAKING UV-ABSORBING OPHTHALMIC LENSES NOVARTIS AG (CH) 2013-04-18 US disclosed
WO-2012015639-A1 METHOD FOR MAKING UV-ABSORBING OPHTHALMIC LENSES NOVARTIS AG (CH) 2012-02-02 WO disclosed
US-20120023869-A1 METHOD FOR MAKING UV-ABSORBING OPHTHALMIC LENSES ALCON INC. (CH) 2012-02-02 US disclosed
US-4874803-A HEAT AND OXIDATION RESISTANCE; PHOTOSTABILITY PENNWALT CORPORATION (US) 1989-10-17 US disclosed
EP-0308886-A2 Dianhydride coupled polymer stabilizers ATOCHEM NORTH AMERICA, INC. (US) 1989-03-29 EP disclosed