SCHEMBL5083791

SCHEMBL5083791

CCN(CC)C(=O)Cc1ccccc1Br

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP3A4 P08684 1/20 0.49
TSHR P16473 2/20 0.46
POLB P06746 1/20 0.44
RIPK1 Q13546 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 2/20 0.42
NFKB1 P19838 1/20 0.42
TSPO P30536 1/20 0.42
LMNA P02545 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ALDH1A1 P00352 2/20 0.42
TAAR1 Q96RJ0 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
BLM P54132 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11029109 0.86 CYP1A2 (0.43) CYP1A2CYP2D6CYP2C19CYP3A4TSHR
SCHEMBL11327583 0.81 TAAR1 (0.48) TSHRRIPK1KMT2ALMNAALDH1A1
SCHEMBL11330969 0.80 TSHR (0.54) TSHRMEN1KMT2AALDH1A1HPGD
SCHEMBL2550830 0.80 AKR1B1 (0.57) CYP1A2CYP2D6CYP2C19CYP3A4POLB
SCHEMBL29944951 0.80 AKR1B1 (0.57) CYP1A2CYP2D6CYP2C19CYP3A4POLB
SCHEMBL11313798 0.79 CYP1A2 (0.49) CYP1A2CYP2D6CYP2C19CYP3A4TSHR
SCHEMBL29379067 0.79 HSD17B10 (0.57) CYP1A2CYP2D6CYP2C19CYP3A4TSHR
SCHEMBL19098912 0.79 CYP1A2 (0.49) CYP1A2CYP2D6CYP2C19CYP3A4MEN1
SCHEMBL11326999 0.76 POLQ (0.61) MEN1KMT2ALMNAALDH1A1TAAR1
SCHEMBL13032640 0.76 TAAR1 (0.43) CYP1A2CYP2D6CYP2C19CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948629-A1 SUBSTITUTED PIPERAZINES AND PIPERIDINES AS MODULATORS OF THE NEUROPEPTIDE Y2 RECEPTOR JANSSEN PHARMACEUTICA N.V. (BE) 2008-07-30 EP disclosed
WO-2007053436-A1 SUBSTITUTED PIPERAZINES AND PIPERIDINES AS MODULATORS OF THE NEUROPEPTIDE Y2 RECEPTOR JANSSEN PHARMACEUTICA N.V. (BE) 2007-05-10 WO disclosed