SCHEMBL5084441

SCHEMBL5084441

COc1ccnc(-c2ncc[nH]2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 2/20 0.44
SMPD3 Q9NY59 1/20 0.41
NISCH Q9Y2I1 2/20 0.41
MTOR P42345 1/20 0.39
ADK P55263 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TXNRD1 Q16881 1/20 0.38
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP19A1 P11511 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
ADRA2A P08913 3/20 0.35
ADRA2C P18825 2/20 0.35
ADRA1D P25100 2/20 0.35
ADRA1A P35348 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24921791 0.76 ALDH1A1 (0.41) ALDH1A1KDM4ESMPD3NISCHMTOR
SCHEMBL20595289 0.73 ALDH1A1 (0.43) ALDH1A1KDM4ESMPD3NISCHMTOR
SCHEMBL5189834 0.73 NISCH (0.42) ALDH1A1KDM4ENISCHMTORADK
SCHEMBL20595284 0.73 NISCH (0.42) ALDH1A1KDM4ENISCHMTORADK
SCHEMBL23370194 0.72 NISCH (0.41) ALDH1A1KDM4ESMPD3NISCHMTOR
SCHEMBL23772037 0.72 NISCH (0.44) ALDH1A1KDM4ESMPD3NISCHMTOR
SCHEMBL24910869 0.72 NISCH (0.41) ALDH1A1KDM4ESMPD3NISCHMTOR
SCHEMBL9026316 0.70 NISCH (0.50) ALDH1A1KDM4ESMPD3NISCHMTOR
SCHEMBL29524578 0.69 KMT2A (0.50) ALDH1A1KDM4EMEN1KMT2ACYP1A2
SCHEMBL15483941 0.69 KMT2A (0.50) ALDH1A1KDM4EMEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008150899-A1 COMBINATION THERAPIES FOR TREATMENT OF CANCER AND INFLAMMATORY DISEASES EMORY UNIVERSITY (US) 2008-12-11 WO claimed
WO-2008150899-A1 COMBINATION THERAPIES FOR TREATMENT OF CANCER AND INFLAMMATORY DISEASES EMORY UNIVERSITY (US) 2008-12-11 WO disclosed