SCHEMBL5085543

SCHEMBL5085543

Cc1c(-c2ccccc2)c(=O)oc2cc(O)cc(Cl)c12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERAP1 Q9NZ08 1/20 0.63
ESR1 P03372 3/20 0.50
ESR2 Q92731 3/20 0.50
ALDH1A1 P00352 6/20 0.49
MAPT P10636 4/20 0.49
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.49
HSP90AA1 P07900 1/20 0.49
KDM4E B2RXH2 4/20 0.48
NPC1 O15118 3/20 0.45
CYP3A4 P08684 3/20 0.45
CYP2C9 P11712 3/20 0.45
CYP2C19 P33261 3/20 0.45
ABCB1 P08183 3/20 0.45
CA12 O43570 2/20 0.45
CYP1A1 P04798 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP19A1 P11511 2/20 0.45
MAOA P21397 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27928272 0.87 ERAP1 (0.64) ERAP1ALDH1A1MAPTKMT2AMEN1
SCHEMBL9755685 0.81 ALDH1A1 (0.63) ERAP1ALDH1A1MAPTKMT2AMEN1
SCHEMBL5326900 0.79 ALDH1A1 (0.60) ERAP1ALDH1A1MAPTKMT2AMEN1
SCHEMBL1608015 0.77 ERAP1 (1.00) ERAP1ESR1ESR2ALDH1A1MAPT
SCHEMBL5431415 0.77 ERAP1 (0.65) ERAP1ESR1ESR2ALDH1A1MAPT
SCHEMBL3079215 0.75 ERAP1 (0.63) ERAP1ESR1ESR2ALDH1A1MAPT
SCHEMBL29038494 0.75 MEN1 (0.63) ERAP1ESR2ALDH1A1MAPTKMT2A
SCHEMBL5425943 0.74 ERAP1 (0.79) ERAP1ESR1ESR2ALDH1A1MAPT
SCHEMBL8118207 0.72 ERAP1 (0.72) ERAP1ALDH1A1MAPTKMT2AMEN1
SCHEMBL14498307 0.72 ALDH1A1 (0.56) ERAP1ESR1ESR2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007115181-A9 COMPOUNDS EXHIBITING EFFLUX INHIBITOR ACTIVITY AND COMPOSITIONS AND USES THEREOF EASTMAN CHEM CO (US) 2008-04-03 WO disclosed
WO-2007115181-A2 COMPOUNDS EXHIBITING EFFLUX INHIBITOR ACTIVITY AND COMPOSITIONS AND USES THEREOF EASTMAN CHEMICAL COMPANY (US) 2007-10-11 WO disclosed