SCHEMBL5086903

SCHEMBL5086903

NC1OCc2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.46
ANPEP P15144 2/20 0.41
CYP2D6 P10635 2/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 1/20 0.40
KDM1A O60341 4/20 0.39
NISCH Q9Y2I1 1/20 0.39
HRH1 P35367 2/20 0.38
RET P07949 1/20 0.38
HTR2C P28335 1/20 0.38
SIGMAR1 Q99720 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
IDO1 P14902 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7229901 0.78 HTR2A (0.44) HTR2ARETRAB9AIDO1
SCHEMBL19829905 0.75 HTR2A (0.41) HTR2AANPEPCYP2D6SLC6A2SLC6A4
SCHEMBL19829949 0.75 HTR2A (0.41) HTR2AANPEPCYP2D6SLC6A2SLC6A4
SCHEMBL19829951 0.75 HTR2A (0.41) HTR2AANPEPCYP2D6SLC6A2SLC6A4
SCHEMBL19835488 0.75 HTR2A (0.41) HTR2AANPEPCYP2D6SLC6A2SLC6A4
SCHEMBL19829904 0.75 HTR2A (0.41) HTR2AANPEPCYP2D6SLC6A2SLC6A4
SCHEMBL19827839 0.75 HTR2A (0.41) HTR2AANPEPCYP2D6SLC6A2SLC6A4
SCHEMBL11397671 0.75 HTR2A (0.41) HTR2AANPEPCYP2D6SLC6A2SLC6A4
SCHEMBL19827837 0.75 HTR2A (0.41) HTR2AANPEPCYP2D6SLC6A2SLC6A4
SCHEMBL117297 0.74 CA9 (0.39) RETNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108368053-A Substituted benzazepine derivatives as antibacterial compounds 葛兰素史密斯克莱知识产权发展有限公司 2018-08-03 CN disclosed
CN-107108596-A The oxazoline compound replaced by fused ring system 巴斯夫欧洲公司 2017-08-29 CN disclosed
CN-103717597-B Heterocyclic compounds as kinase inhibitors 原真股份有限公司 2017-07-04 CN disclosed
CN-106660982-A Histone demethylase inhibitors 赛尔基因昆蒂赛尔研究公司 2017-05-10 CN disclosed
CN-105209452-A 4-amino-6- (heterocyclyl) pyridine-2-carboxylic acid esters and 6-amino-2- (heterocyclyl) pyrimidine-4-carboxylic acid esters and their use as herbicides DOW AGROSCIENCES LLC 2015-12-30 CN disclosed
CN-102803252-A Indole amide derivatives and related compounds for use in the treatment of neurodegenerative diseases UNIV LEUVEN KATH 2012-11-28 CN disclosed
EP-1971595-A2 CETP INHIBITORS Merck & Co., Inc. (US) 2008-09-24 EP disclosed
WO-2007081569-A2 CETP INHIBITORS MERCK & CO., INC. (US) 2007-07-19 WO disclosed