SCHEMBL5090741

SCHEMBL5090741

CC(C)(C)[Si](OCC[C@@H]1OCCc2cc(Br)ccc21)(c1ccccc1)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMYD2 Q9NRG4 3/20 0.38
HTT P42858 2/20 0.36
CYP3A4 P08684 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PTGDR Q13258 1/20 0.34
MAPT P10636 1/20 0.34
HTR1D P28221 4/20 0.33
HTR1A P08908 2/20 0.33
DRD2 P14416 2/20 0.33
DRD4 P21917 2/20 0.33
HTR2A P28223 2/20 0.33
ALDH1A1 P00352 2/20 0.32
TAAR1 Q96RJ0 2/20 0.32
THRB P10828 1/20 0.32
HTR1B P28222 2/20 0.32
KDM4C Q9H3R0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5099018 0.85 SMYD2 (0.37) SMYD2HTTCYP3A4SMN1; SMN2PTGDR
SCHEMBL5093550 0.85 SMYD2 (0.38) SMYD2HTTCYP3A4SMN1; SMN2PTGDR
SCHEMBL5092141 0.84 HTR1D (0.34) HTTMAPTHTR1DHTR1ADRD2
SCHEMBL6811491 0.84 HTR1D (0.34) HTTMAPTHTR1DHTR1ADRD2
SCHEMBL5093614 0.78 SMYD2 (0.38) SMYD2HTTCYP3A4SMN1; SMN2HTR1D
SCHEMBL8554069 0.73 MAPT (0.34) HTTMAPTHTR1DHTR1ADRD2
SCHEMBL1205319 0.73 SMYD2 (0.33) SMYD2HTTCYP3A4SMN1; SMN2HTR1A
SCHEMBL5088651 0.73 HTR1D (0.36) HTTMAPTHTR1DHTR1ADRD2
SCHEMBL6812993 0.73 HTR1D (0.36) HTTMAPTHTR1DHTR1ADRD2
SCHEMBL8549512 0.72 MAPT (0.38) HTTMAPTHTR1DHTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7335660-B2 Isochroman compounds for treatment of CNS disorders ELI LILLY AND COMPANY (US) 2008-02-26 US disclosed
EP-1458703-B1 ISOCHROMAN COMPOUNDS FOR TREATMENT OF CNS DISORDERS LILLY CO ELI (US) 2007-02-28 EP disclosed
US-20050014750-A1 Isochroman compounds for treatment of cns disorders ELI LILLY AND COMPANY 2005-01-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050014750-A1 Isochroman compounds for treatment of cns disorders INA, CNR2, CNR1 SMYD2 928/4885HTT 105/4885CYP3A4 1112/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.