SCHEMBL5097256

SCHEMBL5097256

COC(=O)C1(NC(=O)OC(C)(C)C)CC2(CCC2)C1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.34
MEN1 O00255 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33
PPIA P62937 2/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GHSR Q92847 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
BTK Q06187 1/20 0.31
CTSL P07711 1/20 0.31
DGAT1 O75907 1/20 0.31
GAA P10253 1/20 0.31
HSD11B1 P28845 1/20 0.30
EPHX1 P07099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4094284 0.87 MAPT (0.44) MAPTMEN1MAPK1KMT2APPIA
SCHEMBL5103879 0.86 BTK (0.35) MEN1MAPK1KMT2AL3MBTL1GHSR
SCHEMBL5104037 0.84 KMT2A (0.33) MEN1MAPK1KMT2AGHSRBTK
SCHEMBL1350921 0.83 MAPT (0.47) MAPTMEN1MAPK1KMT2APPIA
SCHEMBL1820679 0.83 MAPT (0.39) MAPTMEN1MAPK1KMT2APPIA
SCHEMBL978565 0.82 MAPT (0.50) MAPTMEN1MAPK1KMT2APPIA
SCHEMBL1353132 0.82 MAPT (0.50) MAPTMEN1MAPK1KMT2APPIA
SCHEMBL22362839 0.81 MEN1 (0.35) MEN1MAPK1KMT2AGHSRCTSL
SCHEMBL28715425 0.81 MEN1 (0.35) MEN1MAPK1KMT2AGHSRDGAT1
SCHEMBL5197158 0.78 MAPT (0.39) MAPTMEN1MAPK1KMT2APPIA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7439263-B2 Pyrrolidine and thiazolidine compounds LES LABORATOIRES SERVIER (FR) 2008-10-21 US disclosed
US-20050261501-A1 Pyrrolidine and thiazolidine compounds LES LABORATOIRES SERVIER (FR) 2005-11-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050261501-A1 Pyrrolidine and thiazolidine compounds DPP4, DPP3, NR4A1 MAPT 4424/4885MEN1 3591/4885MAPK1 3319/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.