SCHEMBL5098258

SCHEMBL5098258

Cc1ccc(C(=O)NC2CC2)cc1-c1ccc(C(=O)Nc2cccc(N3CCN(C)CC3)c2)cc1

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 17/20 0.66
HTR1D P28221 1/20 0.61
HTR1B P28222 1/20 0.61
HTR2A P28223 1/20 0.61
RIPK2 O43353 1/20 0.57
SETD2 Q9BYW2 1/20 0.55
HSPB1 P04792 1/20 0.52
CYP2C9 P11712 1/20 0.52
MAPK11 Q15759 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5102767 0.85 DDR2 (0.66) MAPK14
SCHEMBL5111081 0.82 MAPK1 (0.62) MAPK14RIPK2HSPB1CYP2C9MAPK11
SCHEMBL4703449 0.81 MAPK14 (0.67) MAPK14HTR1DHTR1BHTR2ASETD2
SCHEMBL5106052 0.80 MAPK14 (1.00) MAPK14RIPK2HSPB1CYP2C9MAPK11
SCHEMBL6487595 0.79 MAPK14 (1.00) MAPK14HTR1DHTR1BHTR2AMAPK11
SCHEMBL5110807 0.79 MAPK14 (0.66) MAPK14RIPK2HSPB1CYP2C9MAPK11
SCHEMBL4700916 0.79 MAPK14 (0.67) MAPK14HTR1DHTR1BHTR2ASETD2
SCHEMBL5630096 0.78 MAPK14 (0.87) MAPK14HSPB1CYP2C9MAPK11
SCHEMBL16576384 0.78 MAPK14 (0.64) MAPK14RIPK2HSPB1CYP2C9MAPK11
SCHEMBL5106114 0.76 MAPK14 (0.57) MAPK14RIPK2HSPB1CYP2C9MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7396843-B2 5′-carbamoyl-1,1′-biphenyl-4-carboxamide derivatives and their use as p38 kinase inhibitors GLAXO GROUP LIMITED (GB) 2008-07-08 US disclosed
US-20050038014-A1 5'-carbamoyl-1,1' biphenyl-4-carboxamide derivatives and their use as p38 kinase inhibitors GLAXO GROUP LIMITED (GB) 2005-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050038014-A1 5'-carbamoyl-1,1' biphenyl-4-carboxamide derivatives and their use as p38 kinase inhibitors MAPK1, MAP4K2, MAP3K1 MAPK14 18/4885HTR1D 1243/4885HTR1B 1259/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.